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Epigenetic crosstalk: Pharmacological inhibition of HDACs can rescue defective synaptic morphology and neurotransmission phenotypes associated with loss of the chromatin reader Kismet
Journal article   Peer reviewed

Epigenetic crosstalk: Pharmacological inhibition of HDACs can rescue defective synaptic morphology and neurotransmission phenotypes associated with loss of the chromatin reader Kismet

Nina K. Latcheva, Jennifer M. Viveiros, Edward A. Waddell, Phuong T.T. Nguyen, Faith L.W. Liebl and Daniel R. Marenda
Molecular and cellular neurosciences, v 87
Mar 2018
PMID: 29249293

Abstract

CHARGE syndrome CHD7 Drosophila HDAC HDAC inhibitors Kismet
We are beginning to appreciate the complex mechanisms by which epigenetic proteins control chromatin dynamics to tightly regulate normal development. However, the interaction between these proteins, particularly in the context of neuronal function, remains poorly understood. Here, we demonstrate that the activity of histone deacetylases (HDACs) opposes that of a chromatin remodeling enzyme at the Drosophila neuromuscular junction (NMJ). Pharmacological inhibition of HDAC function reverses loss of function phenotypes associated with Kismet, a chromodomain helicase DNA-binding (CHD) protein. Inhibition of HDACs suppresses motor deficits, overgrowth of the NMJ, and defective neurotransmission associated with loss of Kismet. We hypothesize that Kismet and HDACs may converge on a similar set of target genes in the nervous system. Our results provide further understanding into the complex interactions between epigenetic protein function in vivo. •Pharmacological inhibition of HDAC function suppresses decreased kismet phenotypes.•Our data suggests dynamic interactions between epigenetic readers and erasers.•We hypothesize Kismet and HDAC function antagonistically on same target genes.

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Collaboration types
Domestic collaboration
Web of Science research areas
Neurosciences
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