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Hyperbranched lysine−arginine copolymer for gene delivery
Journal article   Peer reviewed

Hyperbranched lysine−arginine copolymer for gene delivery

Qi Peng, Jianjun Zhu, Yongsheng Yu, Lee Hoffman and Xingkun Yang
Journal of biomaterials science. Polymer ed, v 26(16), pp 1163-1177
02 Nov 2015
PMID: 26249038

Abstract

arginine gene delivery hyperbranched lysine
Based on the reactivity of amine groups and carboxyl groups of L-lysine and L-arginine, thermal polymerization of these two natural amino acids results in hyperbranched lysine-arginine copolymers (P-lys-arg X , where X refers to the relevant molar ratio of arginine to lysine). Hyperbranched polylysine (P-lys) and two derivatives (P-lys-arg 0.10 and P-lys-arg 0.20 ) have been prepared. The arginine-rich hyperbranched polymers can interact with plasmid DNA to form nano-sized particles. The polyplexes were physicochemically analyzed by agarose gel electrophoresis, dynamic light scattering, and zeta potential measurements. Furthermore, their transfection efficiency was assessed, employing COS-7, 293T, and HeLa cell lines. It was found that P-lys showed poorly in its ability of condensation with DNA and transfection efficiency. On the other hand, arginine-rich products resulted to significant enhancement of its transfection efficiency, which is dependent on the content of arginine in the polymers, and the cell line used. P-lys-arg 0.20 exhibited better transfection efficiency under all the condition studied. Besides, P-lys-arg 0.20 showed lower toxicity in COS-7 cells.

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Collaboration types
Domestic collaboration
International collaboration
Web of Science research areas
Engineering, Biomedical
Materials Science, Biomaterials
Polymer Science
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