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Polymorphism at 129 dictates metastable conformations of the human prion protein N-terminal β-sheet
Journal article   Open access

Polymorphism at 129 dictates metastable conformations of the human prion protein N-terminal β-sheet

S. Alexis Paz, Eric Vanden-Eijnden and Cameron F Abrams
Chemical science (Cambridge), v 8(2), pp 1225-1232
2017
PMID: 28451263
url
https://doi.org/10.1039/C6SC03275CView
Published, Version of Record (VoR) Open

Abstract

We study the thermodynamic stability of the native state of the human prion protein using a new free-energy method, replica-exchange on-the-fly parameterization. This method is designed to overcome hidden-variable sampling limitations to yield nearly error-free free-energy profiles along a conformational coordinate. We confirm that all four (M129V, D178N) polymorphs have a ground-state conformation with three intact β-sheet hydrogen bonds. Additionally, they are observed to have distinct metastabilities determined by the side-chain at position 129. We rationalize these findings with reference to the prion “strain” hypothesis, which links the variety of transmissible spongiform encephalopathy phenotypes to conformationally distinct infectious prion forms and classifies distinct phenotypes of sporadic Creutzfeldt-Jakob disease based solely on the 129 polymorphism. Because such metastable structures are not easily observed in structural experiments, our approach could potentially provide new insights into the conformational origins of prion diseases and other pathologies arising from protein misfolding and aggregation.

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Collaboration types
Domestic collaboration
Web of Science research areas
Chemistry, Multidisciplinary
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