Logo image
Synthesis of (2 R, 3 S)-methyl-2-fluoro-3-(n-benzoylamino)-3-phenylpropanoate: Modified side chain of taxol
Journal article   Peer reviewed

Synthesis of (2 R, 3 S)-methyl-2-fluoro-3-(n-benzoylamino)-3-phenylpropanoate: Modified side chain of taxol

Franklin A. Davis and Rajarathnam E. Reddy
Tetrahedron: asymmetry, v 5(6), pp 955-960
1994

Abstract

Methyl-2-fluoro-3-(N-benzoylamino)-3-phenylpropanoate 2 and 3, fluorine analogs of the C-13 side chain of taxol, were synthesized by electrophilic fluorination of the dianion of methyl ( R)-(−)-(N-benzoyl)-3-amino-3-phenylpropanoale ( 4). Methyl-2-fluoro-3-(N-benzoylamino)-3-phenylpropanoate 2 and 3, fluorine analogs of the C-13 side chain of taxol, were synthesized by electrophilic fluorination of the dianion of methyl ( R)-(−)-benzoyl)-3-amino-3-phenylpropanoate ( 4) with NFOBS 6.

Metrics

9 Record Views
46 citations in Scopus

Details

UN Sustainable Development Goals (SDGs)

This publication has contributed to the advancement of the following goals:

#3 Good Health and Well-Being
#13 Climate Action

InCites Highlights

Data related to this publication, from InCites Benchmarking & Analytics tool:

Web of Science research areas
Chemistry, Inorganic & Nuclear
Chemistry, Organic
Chemistry, Physical
Logo image